《活性多肽与药物开发》

《活性多肽与药物开发》
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绵乖石钸尔;乖毋乖秘不尔也不!矫茚!绵’矫茚尔尔’!{‘乖
~--tS预告?
《活性多肽与药物开发》
王德心着
中国医药科技出版社2008年7月出版
全书共134.5万字,分上篇总论及下篇各论.
上篇内容为肽的特性,分类,剂型,合成策略,巧妙合成例.针对经典肽的修饰与改造是本篇的重点.
其中包括伪肽,环肽,Fridinger肽,简化肽及加合肽,拟肽等主要类型的合成方法,还包括开发为新先导物
药物的实例.
下篇内容按不同生物活性分别介绍了抗肿瘤肽,免疫活性肽,镇痛肽,造血活性肽,骨代谢肽,神经活
性肽,抗生素肽,生长及血糖调节肽,抗凝肽,核素标记肽,合成肽疫苗,蛋白酶结合肽等内容.
文中配合大量的合成反应,目标结构图示及充分的文献是该书的另一特点.。