常见药物中间体

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常见药物中间体

Entecavir恩替卡韦中间体:

第1步:

3-Cyclopenten-1-ol,2-[(phenylmethoxy)methyl]-,(1R-trans) CAS No:188399-48-6

第2步:

(1S,2R,3S,5R)-2-(benzyloxymethyl)-6-oxabicyclo[3.1.0]hexan-3-ol CAS No:117641-39-1 第3步:

6-Oxabicyclo[3.1.0]hexane,3-(phenylmethoxy)-2-[(phenylmethoxy)methyl]-, (1S,2R,3S,5R) CAS No 110567-22-1

第4步:

(1S,2S,3S,5S)-5-(2-amino-6-(benzyloxy)-9H-purin-9-yl)-3-(benzyloxy)-2- (benzyloxymethyl)cyclopentanol

cas:142217-77-4

第5步:

(2R,3S,5S)-3-(benzyloxy)-5-(6-(benzyloxy)-2- ((4-methoxyphenyl)diphenylmethylamino)- 9H-purin-9-yl)-2-(benzyloxymethyl)cyclopentanol CAS No:142217-78-5

第6步:

(2R,3S,5S)-3-(benzyloxy)-5-(6-(benzyloxy)-2-((4-methoxyphenyl) diphenylmethylamino)-9H-purin-9-yl)-2-(benzyloxymethyl)cyclopentanone CAS No 142217-79-6

第7步:

6-(benzyloxy)-9-((1S,3R,4S)-4-(benzyloxy)-3-(benzyloxymethyl)-2

-methylenecyclopentyl)-N-((4-methoxyphenyl)diphenylmethyl) -9H-purin-2-amine CAS No 142217-80-9

第8步:

6-(benzyloxy)-9-((1S,3R,4S)-4-(benzyloxy)-3-(benzyloxymethyl)-2- methylenecyclopentyl)-9H-purin-2-amine CAS No 204845-95-4

钆双胺一水物122795-43-1

阿折地平中间体

阿折地平中间体 CAS:18621-17-5

阿折地平中间体 CAS:116574-14-2

阿折地平中间体 CAS:170749-59-4

阿折地平中间体 CAS:39562-25-9

Anagrelide阿那格雷中间体

N-(6-硝基-2.3-二氯苄基)甘氨酸乙酯盐酸盐

N-(2.3-dichloro-6-nitrobenzyl)glycine HCl 含量:98%以上 99%

N-(6-氨基-2.3-二氯苄基)甘氨酸乙酯

Ethyl N-(6-amino-2.3-dichlorobenzyl)glycine 70406-92-7

Prasugrel普拉格雷侧链(中间体)150322-73-9 含量:98%以上

Adapalene 阿达帕林中间体:

2-(1-Adamantyl)-4-bromophenol

2-(1-金刚烷基)-4-溴苯酚

2-(1-Adamantyl)-4-bromoanisole

2-(1-金刚烷基)-4-溴苯甲醚

Methyl 6-[3-(1-adamantyl)-4-methoxyphenyl]-2-naphthoate

6-[3-(1-金刚烷基)-4-甲氧基苯基]-2-萘甲酸甲酯

1-(5-Bromo-2-Methoxyphenyl)-adamantane CAS NO.104224-63-7 1-(5-溴-2-甲氧基苯基)金刚烷

Methyl 6-bromo-2-naphthoate

6-溴-2-萘甲酸甲酯

Adefovir Dipivoxil 阿徳福韦酯中间体:

9-[2-(Diethylphosphonomethoxy)ethyl]adenine

9-[2-(二乙基膦酸基甲氧基)乙基]腺嘌呤

9-(2-Phosphonylmethoxyethyl]adenine(Adefovir)

9-[2-(膦酸基甲氧基)乙基]腺嘌呤(阿德福韦)

Amorolfine HCl 盐酸阿莫罗芬中间体:

3-[1,1-Dimethylphenyl-4-]-2-methyl-propionic acid

3-[1,1-二甲基苯基-4-]-2-甲基-丙酸

Anagrelide 阿那格雷中间体:

Ethyl N-(2,3-dichloro-6-amino benzyl)glycine

N-(2,3-二氯-6-氨基-苄基)甘氨酸乙酯

Aripiprazole阿立哌唑中间体:

1-(2,3-Dichloro-phenyl)-piperazine hydrobromide

1-(2,3-二氯苯基)-哌嗪氢溴酸盐

7-(4-Bromo-butoxy)-3,4-dihydro-2(1H)-quinolinone

7-(4-溴丁氧基)-3,4-二氢-2(1H)-喹啉酮

Brompheniramine Maleate马来酸溴苯那敏中间体:

α-(p-Bromophenyl)-α-(β-dimethylaminoethyl)-2-pyridylacetonitrile maleate

α-对溴苯基-α-(β-二甲基氨基乙基)-2-吡啶乙腈马来酸盐

Candesartan Cilexetil 坎地沙坦酯中间体:

Cyclohexyl 1-chloroethylcarbonate

环己基1-氯乙基碳酸酯

2-Ethoxy-1-[[2’-(1H-tetrezol-5-yl)biphenyl-4-yl]-methyl]benzimidazole-7-carboxylic acid (Candesartan)

1-[[2'-(1-H-四氮唑-5-基)联苯-4-基]甲基]-2-乙氧基-苯并咪唑-7-羧酸(坎地沙坦)

Cefepime头孢吡肟中间体:

(6R, 7R)-7-Amino-3-[(1-methyl-1-pyrrolidino)methyl]ceph-3-em-4-carboxylate hydriodic acid 7-氨基-3-[(1-甲基-1-吡咯烷基)甲基]头孢-3-烯基-4-羧基氢碘酸盐(头孢吡肟母核)

Cefutibuten 头孢布烯中间体:

(E/Z) (4-2-Methyl-buten) 4-(2-benzyloxycarbonyolaminothiazol-4-yl)-4-carboxy-3-butyrate (Cefutibuten side chain)

(顺/反)4-(2-苄氧羰基氨基噻唑-4-基)-4-羧基-3-丁烯酸(4-2-甲基-2-丁烯)酯(头孢布烯侧链)

Dofetilide 多非利特中间体:

2-[4-Nitrophenoxy]ethyl chloride

4-(2-氯乙氧基)硝基苯

N-Methyl-4-nitrophenethylamine hydrochloride CAS: 166943-39-1

4-硝基-β-苯乙胺盐酸盐

N-Methyl-N-[2-(4-nitrophenoxy)ethyl]-4-nitrophenylamine

N-甲基-N-[2-(4-硝基苯氧基)乙基]-4-硝基苯乙胺

Escitalopram Oxalate草酸依地普仑中间体:

(-)-4-[4-(Dimethylamino)-1-(4’-fluorophenyl)-1-hydroxy-1-butyl]-3-(hydroxymethyl)benzonitrile, Tosyltartaric acid salt

(-)-4-[4-二甲氨基-1-(4-氟苯基)-1-羟基-1-丁基]-3-羟甲基苯乙腈,苯甲酰基酒石酸盐Finasteride非那雄胺中间体:

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